DE FRANCO, MICHELE
DE FRANCO, MICHELE
Dipartimento di Scienze del Farmaco - DSF
1,3,5-Triaza-7-phosphaadamantane and Cyclohexyl Groups Impart to Di-Iron(I) Complex Aqueous Solubility and Stability, and Prominent Anticancer Activity in Cellular and Animal Models
2024 De Franco, M.; Biancalana, L.; Zappelli, C.; Zacchini, S.; Gandin, V.; Marchetti, F.
Anticancer activity of new water-soluble sulfonated thiosemicarbazone copper(II) complexes targeting disulfide isomerase
2024 Miglioli, F.; De Franco, M.; Bartoli, J.; Scaccaglia, M.; Pelosi, G.; Marzano, C.; Rogolino, D.; Gandin, V.; Carcelli, M.
DEVELOPMENT OF TARGET-SPECIFIC AND TUMOR-SELECTIVE METALLODRUGS
2024 DE FRANCO, Michele
Synthesis, characterization and in vitro cytotoxicity of gallium(iii)-dithiocarbamate complexes
2024 Salvarese, N.; Morellato, N.; Gobbi, C.; Gandin, V.; De Franco, M.; Marzano, C.; Dolmella, A.; Bolzati, C.
Triiron Complex with N-Ferrocenyl Aminocarbyne Ligand Bridging a Diiron Core: DFT, Electrochemical, and Biological Insights
2024 Saviozzi, Chiara; Biancalana, Lorenzo; Funaioli, Tiziana; Bortoluzzi, Marco; De Franco, Michele; Guelfi, Massimo; Gandin, Valentina; Marchetti, Fabio
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
2023 Pecoraro, Camilla; DE FRANCO, Michele; Carbone, Daniela; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall'Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; DE FRANCO, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Novel Biotinylated Cu(II)-Phenanthroline Complexes: 2D and 3D Cytotoxic Activity and Mechanistic Insight
2023 Barrett, Stephen; De Franco, Michele; Donati, Chiara; Marzano, Cristina; Gandin, Valentina; Montagner, Diego
Novel Silver Complexes Based on Phosphanes and Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands Targeting TrxR: New Promising Chemotherapeutic Tools Relevant to SCLC Management
2023 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Caviglia, Miriam; Sgarbossa, Paolo; De Franco, Michele; Zancato, Mirella; Marzano, Cristina; Gandin, Valentina
Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; De Franco, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Sut, Stefania; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Unusual tellurium(iv) mediated cyclisation diols into dihydroxazoles with potential anticancer activity
2023 D’Arcy, Kenneth; Schäfer, Tim; De Franco, Michele; Ricco, Raffaele; Gandin, Valentina; Sanz Miguel, Pablo J.; Montagner, Diego
Cu(I) and Cu(II) Complexes Based on Lonidamine-Conjugated Ligands Designed to Promote Synergistic Antitumor Effects
2022 Del Bello, Fabio; Pellei, Maura; Bagnarelli, Luca; Santini, Carlo; Giorgioni, Gianfabio; Piergentili, Alessandro; Quaglia, Wilma; Battocchio, Chiara; Iucci, Giovanna; Schiesaro, Irene; Meneghini, Carlo; Venditti, Iole; Ramanan, Nitya; De Franco, Michele; Sgarbossa, Paolo; Marzano, Cristina; Gandin, Valentina
Decoding mechanism of action and sensitivity to drug candidates from integrated transcriptome and chromatin state
2022 Carraro, Caterina; Bonaguro, Lorenzo; Schulte-Schrepping, Jonas; Horne, Arik; Oestreich, Marie; Warnat-Herresthal, Stefanie; Helbing, Tim; De Franco, Michele; Haendler, Kristian; Mukherjee, Sach; Ulas, Thomas; Gandin, Valentina; Goettlich, Richard; Aschenbrenner, Anna C; Schultze, Joachim L; Gatto, Barbara
Exploring the Antitumor Potential of Copper Complexes Based on Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands
2022 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Battocchio, Chiara; Iucci, Giovanna; Venditti, Iole; Meneghini, Carlo; Amatori, Simone; Sgarbossa, Paolo; Marzano, Cristina; De Franco, Michele; Gandin, Valentina
Insight on pyrimido[5,4-g]indolizine and pyrimido[4,5-c]pyrrolo[1,2-a]azepine systems as promising photosensitizers on malignant cells
2022 Barreca, M; Ingarra, Am; Raimondi, Mv; Spanò, V; De Franco, M; Menilli, L; Gandin, V; Miolo, G; Barraja, P; Montalbano, A.
New tricyclic systems as photosensitizers towards triple negative breast cancer cells
2022 Barreca, Marilia; Ingarra, Angela Maria; Raimondi, Maria Valeria; Spanò, Virginia; Piccionello, Antonio Palumbo; De Franco, Michele; Menilli, Luca; Gandin, Valentina; Miolo, Giorgia; Barraja, Paola; Montalbano, Alessandra
Preliminary Discovery of Small Molecule Inhibitors of Epidermal Growth Factor Receptor (EGFR) That Bind to the Extracellular Domain
2022 Di Liddo, Rosa; Verona, Marco; Vaccarin, Christian; Acquasaliente, Laura; Schrenk, Sandra; Piccione, Monica; Cenzi, Carola; De Franco, Michele; Dal Prà, Matteo; Ribaudo, Giovanni; Ferlin, Maria Grazia; Conconi, Maria Teresa; Chilin, Adriana; Gandin, Valentina; Marzaro, Giovanni
Unveiling the Potential of Innovative Gold(I) and Silver(I) Selenourea Complexes as Anticancer Agents Targeting TrxR and Cellular Redox Homeostasis
2022 De Franco, Michele; Saab, Marina; Porchia, Marina; Marzano, Cristina; Nolan, Steven P; Nahra, Fady; Van Hecke, Kristof; Gandin, Valentina
Appended Aromatic Moieties in Flexible Bis‐3‐chloropiperidines Confer Tropism against Pancreatic Cancer Cells
2021 Carraro, Caterina; Helbing, Tim; Francke, Alexander; Zuravka, Ivonne; Sosic, Alice; De Franco, Michele; Gandin, Valentina; Gatto, Barbara; Göttlich, D. Richard
Easily Available, Amphiphilic Diiron Cyclopentadienyl Complexes Exhibit in Vitro Anticancer Activity in 2D and 3D Human Cancer Cells through Redox Modulation Triggered by CO Release
2021 Biancalana, L.; De Franco, M.; Ciancaleoni, G.; Zacchini, S.; Pampaloni, G.; Gandin, V.; Marchetti, F.