MARZARO, GIOVANNI
MARZARO, GIOVANNI
Dipartimento di Scienze del Farmaco - DSF
Discovery of selective, metabolically stable pyrazole-based FLT3 inhibitors for the treatment of acute myeloid leukemia
2025 Destro, L.; Crippa, V.; Gabbia, D.; Roverso, M.; Bogialli, S.; Zardi, P.; Marzaro, G.; Mologni, L.; Zambon, A.
Aged Garlic Extract (AGE) and Its Constituent S-Allyl-Cysteine (SAC) Inhibit the Expression of Pro-Inflammatory Genes Induced in Bronchial Epithelial IB3-1 Cells by Exposure to the SARS-CoV-2 Spike Protein and the BNT162b2 Vaccine
2024 Gasparello, J.; Papi, C.; Marzaro, G.; Macone, A.; Zurlo, M.; Finotti, A.; Agostinelli, E.; Gambari, R.
Biodistribution Assessment of a Novel 68Ga-Labeled Radiopharmaceutical in a Cancer Overexpressing CCK2R Mouse Model: Conventional and Radiomics Methods for Analysis
2024 Maria Pavone, Anna; Benfante, Viviana; Giaccone, Paolo; Stefano, Alessandro; Torrisi, Filippo; Russo, Vincenzo; Serafini, Davide; Richiusa, Selene; Pometti, Marco; Scopelliti, Fabrizio; Ippolito, Massimo; Giulio Giannone, Antonino; Cabibi, Daniela; Asti, Mattia; Vettorato, Elisa; Morselli, Luca; Merone, Mario; Lunardon, Marcello; Andrighetto, Alberto; Tuttolomondo, Antonino; Paolo Cammarata, Francesco; Verona, Marco; Marzaro, Giovanni; Mastrotto, Francesca; Parenti, Rosalba; Russo, Giorgio; Comelli, Albert
Deformable Vesicles with Edge Activators for the Transdermal Delivery of Non-Psychoactive Cannabinoids
2024 Vettorato, Elisa; Fiordelisi, Marisa; Ferro, Silvia; Zanin, Desirè; Franceschinis, Erica; Marzaro, Giovanni; Realdon, Nicola
Development and Validation of Novel Z-360-Based Macromolecules for the Active Targeting of CCK2-R
2024 Vettorato, E.; Verona, M.; Bellio, G.; Croci, S.; Filadi, R.; Bisio, A.; Spessot, E.; Andrighetto, A.; Maniglio, D.; Asti, M.; Marzaro, G.; Mastrotto, F.
Synthesis and Biological Evaluation of Pyrazole-Pyrimidones as a New Class of Correctors of the Cystic Fibrosis Transmembrane Conductance Regulator (CFTR)
2024 Vaccarin, Christian; Veit, Guido; Hegedus, Tamas; Torres, Odalys; Chilin, Adriana; Lukacs, Gergely L; Marzaro, Giovanni
Assessing the interaction between hemoglobin and the receptor binding domain of SARS-CoV-2 spike protein through MARTINI coarse-grained molecular dynamics
2023 Gasparello, J.; Verona, M.; Chilin, A.; Gambari, R.; Marzaro, G.
Effects of Sulforaphane on SARS‑CoV‑2 infection and NF‑κB dependent expression of genes involved in the COVID‑19 ‘cytokine storm’
2023 Gasparello, J.; Marzaro, G.; Papi, C.; Gentili, V.; Rizzo, R.; Zurlo, M.; Scapoli, C.; Finotti, A.; Gambari, R.
Inhibitory effects of SARS-CoV-2 spike protein and BNT162b2 vaccine on erythropoietin-induced globin gene expression in erythroid precursor cells from patients with β-thalassemia
2023 Cosenza, L. C.; Marzaro, G.; Zurlo, M.; Gasparello, J.; Zuccato, C.; Finotti, A.; Gambari, R.
The anti-SARS-CoV-2 BNT162b2 vaccine suppresses mithramycin-induced erythroid differentiation and expression of embryo-fetal globin genes in human erythroleukemia K562 cells
2023 Zurlo, M.; Gasparello, J.; Verona, M.; Papi, C.; Cosenza, L. C.; Finotti, A.; Marzaro, G.; Gambari, R.
A NEW PRODUCTION METHOD OF HIGH SPECIFIC ACTIVITY RADIONUCLIDES TOWARDS INNOVATIVE RADIOPHARMACEUTICALS: THE ISOLPHARM PROJECT
2022 Vettorato, E.; Morselli, L.; Ballan, M.; Arzenton, A.; Khwairakpam, O. S.; Verona, M.; Scarpa, D.; Corradetti, S.; Caliceti, P.; Di Marco, V.; Mastrotto, F.; Marzaro, G.; Realdon, N.; Zenoni, A.; Donzella, A.; Lunardon, M.; Zangrando, L.; Asti, M.; Russo, G.; Mariotti, E.; Maniglio, D.; Andrighetto, A.
A novel phenolic derivative inhibits AHL-dependent Quorum Sensing signaling in Pseudomonas aeruginosa
2022 Bernabè, Giulia; Marzaro, Giovanni; DI PIETRA, Giuseppe; Otero, Ana; Bellato, Massimo; Pauletto, Anthony; Scarpa, Melania; Sut, Stefania; Chilin, Adriana; Dall’Acqua, Stefano; Brun, Paola; Castagliuolo, Ignazio
Improved Trimethylangelicin Analogs for Cystic Fibrosis: Design, Synthesis and Preliminary Screening
2022 Vaccarin, Christian; Gabbia, Daniela; DE MARTIN, Sara; Franceschinis, Erica; Roverso, Marco; Bogialli, Sara; Sacchetti, Gianni; Lampronti, Ilaria; Cabrini, Giulio; Cristina Dechecchi, Maria; Tamanini, Anna; Marzaro, Giovanni; Chilin, Adriana
Preliminary Discovery of Small Molecule Inhibitors of Epidermal Growth Factor Receptor (EGFR) That Bind to the Extracellular Domain
2022 Di Liddo, Rosa; Verona, Marco; Vaccarin, Christian; Acquasaliente, Laura; Schrenk, Sandra; Piccione, Monica; Cenzi, Carola; De Franco, Michele; Dal Prà, Matteo; Ribaudo, Giovanni; Ferlin, Maria Grazia; Conconi, Maria Teresa; Chilin, Adriana; Gandin, Valentina; Marzaro, Giovanni
Proteolysis Targeting Chimeric Molecules: Tuning Molecular Strategies for a Clinically Sound Listening
2022 Pedrucci, Federica; Pappalardo, Claudia; Marzaro, Giovanni; Ferri, Nicola; Ferlin, Alberto; DE TONI, Luca
A Novel Aza-Derivative Inhibits agr Quorum Sensing Signaling and Synergizes Methicillin-Resistant Staphylococcus aureus to Clindamycin
2021 Bernabe, G.; Dal Pra, M.; Ronca, V.; Pauletto, A.; Marzaro, G.; Saluzzo, F.; Stefani, ANNA-LISA; Artusi, I.; De Filippis, V.; Ferlin, M. G.; Brun, P.; Castagliuolo, I.
Dual kinase targeting in leukemia
2021 Mologni, L.; Marzaro, G.; Redaelli, S.; Zambon, A.
Preliminary Study of a 1,5-Benzodiazepine-Derivative Labelled with Indium-111 for CCK-2 Receptor Targeting
2021 Verona, Marco; Rubagotti, Sara; Croci, Stefania; Sarpaki, Sophia; Borgna, Francesca; Tosato, Marianna; Vettorato, Elisa; Marzaro, Giovanni; Mastrotto, Francesca; Asti, Mattia
Tyrosine kinase inhibitor prodrug-loaded liposomes for controlled release at tumor microenvironment
2021 Salmaso, S.; Mastrotto, F.; Roverso, M.; Gandin, V.; De Martin, S.; Gabbia, D.; De Franco, M.; Vaccarin, C.; Verona, M.; Chilin, A.; Caliceti, P.; Bogialli, S.; Marzaro, G.
Preliminary evaluation of the production of non-carrier added 111Ag as core of a therapeutic radiopharmaceutical in the framework of ISOLPHARM_Ag experiment
2020 Ballan, Michele; Tosato, Marianna; Verona, Marco; Caeran, Michele; Borgna, Francesca; Vettorato, Elisa; Corradetti, Stefano; Zangrando, Lisa; Sgaravatto, Massimo; Verlato, Marco; Asti, Mattia; Marzaro, Giovanni; Mastrotto, Francesca; Di Marco, Valerio; Maniglio, Devid; Bisio, Alessandra; Motta, Antonella; Quaranta, Alberto; Zenoni, Aldo; Pastore, Paolo; Realdon, Nicola; Andrighetto, Alberto