SALMASO, VERONICA
SALMASO, VERONICA
Dipartimento di Scienze del Farmaco - DSF
7-Amino-[1,2,4]triazolo[1,5-a][1,3,5]triazines as CK1δ inhibitors: Exploring substitutions at the 2 and 5-positions
2024 Grieco, Ilenia; Bassani, Davide; Trevisan, Letizia; Salmaso, Veronica; Cescon, Eleonora; Prencipe, Filippo; Da Ros, Tatiana; Martinez-Gonzalez, Loreto; Martinez, Ana; Spalluto, Giampiero; Moro, Stefano; Federico, Stephanie
A second life for the crystallographic structure of Berenil-dodecanucleotide complex: a computational revisitation thirty years after its publication
2024 Novello, Gianluca; Dodaro, Andrea; Menin, Silvia; Cavastracci Strascia, Chiara; Sturlese, Mattia; Salmaso, Veronica; Moro, Stefano
Extrahelical Binding Site for a 1H-Imidazo[4,5-c]quinolin-4-amine A3Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7
2024 Fisher, Courtney L.; Pavan, Matteo; Salmaso, Veronica; Keyes, Robert F.; Wan, Tina C.; Pradhan, Balaram; Gao, Zhan-Guo; Smith, Brian C.; Jacobson, Kenneth A.; Auchampach, John A.
Lipid Trolling to Optimize A3 Adenosine Receptor-Positive Allosteric Modulators (PAMs)
2024 Pradhan, Balaram; Pavan, Matteo; Fisher, Courtney L.; Salmaso, Veronica; Wan, Tina C.; Keyes, Robert F.; Rollison, Noah; Suresh, R. Rama; Kumar, T. Santhosh; Gao, Zhan-Guo; Smith, Brian C.; Auchampach, John A.; Jacobson, Kenneth A.
Photoswitchable Diazocine Derivative for Adenosine A3 Receptor Activation in Psoriasis
2024 López-Cano, Marc; Scortichini, Mirko; Tosh, Dilip K.; Salmaso, Veronica; Ko, Tongil; Salort, Glòria; Filgaira, Ingrid; Soler, Concepció; Trauner, Dirk; Hernando, Jordi; Jacobson, Kenneth A.; Ciruela, Francisco
Stereocontrolled access to thioisosteres of nucleoside di- and triphosphates
2024 Zhang, Hai-Jun; Ociepa, Michał; Nassir, Molhm; Zheng, Bin; Lewicki, Sarah A.; Salmaso, Veronica; Baburi, Helay; Nagel, Jessica; Mirza, Salahuddin; Bueschbell, Beatriz; Al-Hroub, Haneen; Perzanowska, Olga; Lin, Ziqin; Schmidt, Michael A.; Eastgate, Martin D.; Jacobson, Kenneth A.; Müller, Christa E.; Kowalska, Joanna; Jemielity, Jacek; Baran, Phil S.
Structural Investigations on 2-Amidobenzimidazole Derivatives as New Inhibitors of Protein Kinase CK1 Delta
2024 Calenda, Sara; Catarzi, Daniela; Varano, Flavia; Vigiani, Erica; Volpini, Rosaria; Lambertucci, Catia; Spinaci, Andrea; Trevisan, Letizia; Grieco, Ilenia; Federico, Stephanie; Spalluto, Giampiero; Novello, Gianluca; Salmaso, Veronica; Moro, Stefano; Colotta, Vittoria
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
2023 Oliva, Paola; Suresh, R. Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J.; Tosh, Dilip K.; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A.
[1,2,4]Triazolo[1,5‐c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines
2023 Federico, Stephanie; Persico, Margherita; Trevisan, Letizia; Biasinutto, Chiara; Bolcato, Giovanni; Salmaso, Veronica; Da Ros, Tatiana; Gianferrara, Teresa; Prencipe, Filippo; Kachler, Sonja; Klotz, Karl‐norbert; Pacor, Sabrina; Moro, Stefano; Spalluto, Giampiero
First Potent Macrocyclic A3 Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences
2023 Tosh, Dilip K.; Fisher, Courtney L.; Salmaso, Veronica; Wan, Tina C.; Campbell, Ryan G.; Chen, Eric; Gao, Zhan-Guo; Auchampach, John A.; Jacobson, Kenneth A.
Fluorescent A2A and A3 adenosine receptor antagonists as flow cytometry probes
2023 Toti, Kiran S; Campbell, Ryan G; Lee, Hobin; Salmaso, Veronica; Suresh, R Rama; Gao, Zhan-Guo; Jacobson, Kenneth A
Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors
2023 Salmaso, Veronica; Persico, Margherita; Da Ros, Tatiana; Spalluto, Giampiero; Kachler, Sonja; Klotz, Karl-Norbert; Moro, Stefano; Federico, Stephanie
Thermal Titration Molecular Dynamics (TTMD): Not Your Usual Post-Docking Refinement
2023 Menin, Silvia; Pavan, Matteo; Salmaso, Veronica; Sturlese, Mattia; Moro, Stefano
Thermal titration molecular dynamics (TTMD): shedding light on the stability of RNA-small molecule complexes
2023 Dodaro, Andrea; Pavan, Matteo; Menin, Silvia; Salmaso, Veronica; Sturlese, Mattia; Moro, Stefano
A3 adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity
2022 Tosh, Dilip K; Salmaso, Veronica; Campbell, Ryan G; Rao, Harsha; Bitant, Amelia; Pottie, Eline; Stove, Christophe P; Liu, Naili; Gavrilova, Oksana; Gao, Zhan-Guo; Auchampach, John A; Jacobson, Kenneth A
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist
2022 Wen, Zhiwei; Salmaso, Veronica; Jung, Young-Hwan; Phung, Ngan B; Gopinatth, Varun; Shah, Qasim; Patterson, Alexandra T; Randle, John C R; Chen, Zhoumou; Salvemini, Daniela; Lieberman, David I; Whitehead, Gregory S; Karcz, Tadeusz P; Cook, Donald N; Jacobson, Kenneth A
Selective A3 Adenosine Receptor Antagonist Radioligand for Human and Rodent Species
2022 Suresh, R Rama; Gao, Zhan-Guo; Salmaso, Veronica; Chen, Eric; Campbell, Ryan G; Poe, Russell B; Liston, Theodore E; Jacobson, Kenneth A
Structure-Activity Relationship of 3-Methylcytidine-5'-α,β-methylenediphosphates as CD73 Inhibitors
2022 Scortichini, Mirko; Idris, Riham Mohammed; Moschütz, Susanne; Keim, Antje; Salmaso, Veronica; Dobelmann, Clemens; Oliva, Paola; Losenkova, Karolina; Irjala, Heikki; Vaittinen, Samuli; Sandholm, Jouko; Yegutkin, Gennady G; Sträter, Norbert; Junker, Anna; Müller, Christa E; Jacobson, Kenneth A
Structure-Activity Studies of 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as A3 Adenosine Receptor Positive Allosteric Modulators
2022 Fallot, Lucas B; Suresh, R Rama; Fisher, Courtney L; Salmaso, Veronica; O'Connor, Robert D; Kaufman, Noy; Gao, Zhan-Guo; Auchampach, John A; Jacobson, Kenneth A
Synthesis and Effect of Conformationally Locked Carbocyclic Guanine Nucleotides on Dynamin
2022 Toti, Kiran S; Jimah, John R; Salmaso, Veronica; Hinshaw, Jenny E; Jacobson, Kenneth A