CHILIN, ADRIANA
CHILIN, ADRIANA
Dipartimento di Scienze del Farmaco - DSF
Synthesis and Biological Evaluation of Pyrazole-Pyrimidones as a New Class of Correctors of the Cystic Fibrosis Transmembrane Conductance Regulator (CFTR)
2024 Vaccarin, Christian; Veit, Guido; Hegedus, Tamas; Torres, Odalys; Chilin, Adriana; Lukacs, Gergely L; Marzaro, Giovanni
Assessing the interaction between hemoglobin and the receptor binding domain of SARS-CoV-2 spike protein through MARTINI coarse-grained molecular dynamics
2023 Gasparello, J.; Verona, M.; Chilin, A.; Gambari, R.; Marzaro, G.
A novel phenolic derivative inhibits AHL-dependent Quorum Sensing signaling in Pseudomonas aeruginosa
2022 Bernabè, Giulia; Marzaro, Giovanni; DI PIETRA, Giuseppe; Otero, Ana; Bellato, Massimo; Pauletto, Anthony; Scarpa, Melania; Sut, Stefania; Chilin, Adriana; Dall’Acqua, Stefano; Brun, Paola; Castagliuolo, Ignazio
Emergent treatments for β-thalassemia and orphan drug legislations
2022 Costa, Enrico; Domenica Cappellini, Maria; Rivella, Stefano; Chilin, Adriana; Alessi, Eva; Riccaboni, Massimo; Leufkens, Hubert G M; Luzzatto, Lucio
Improved Trimethylangelicin Analogs for Cystic Fibrosis: Design, Synthesis and Preliminary Screening
2022 Vaccarin, Christian; Gabbia, Daniela; DE MARTIN, Sara; Franceschinis, Erica; Roverso, Marco; Bogialli, Sara; Sacchetti, Gianni; Lampronti, Ilaria; Cabrini, Giulio; Cristina Dechecchi, Maria; Tamanini, Anna; Marzaro, Giovanni; Chilin, Adriana
New TMA (4,6,4'-Trimethyl angelicin) Analogues as Anti-Inflammatory Agents in the Treatment of Cystic Fibrosis Lung Disease
2022 Tupini, Chiara; Chilin, Adriana; Rossi, Alice; De Fino, Ida; Bragonzi, Alessandra; D'Aversa, Elisabetta; Cosenza, Lucia Carmela; Vaccarin, Christian; Sacchetti, Gianni; Borgatti, Monica; Tamanini, Anna; Dechecchi, Maria Cristina; Sanvito, Francesca; Gambari, Roberto; Cabrini, Giulio; Lampronti, Ilaria
Preliminary Discovery of Small Molecule Inhibitors of Epidermal Growth Factor Receptor (EGFR) That Bind to the Extracellular Domain
2022 Di Liddo, Rosa; Verona, Marco; Vaccarin, Christian; Acquasaliente, Laura; Schrenk, Sandra; Piccione, Monica; Cenzi, Carola; De Franco, Michele; Dal Prà, Matteo; Ribaudo, Giovanni; Ferlin, Maria Grazia; Conconi, Maria Teresa; Chilin, Adriana; Gandin, Valentina; Marzaro, Giovanni
Self-Emulsifying Formulations to Increase the Oral Bioavailability of 4,6,4′-Trimethylangelicin as a Possible Treatment for Cystic Fibrosis
2022 Franceschinis, Erica; Roverso, Marco; Gabbia, Daniela; De Martin, Sara; Brusegan, Matteo; Vaccarin, Christian; Bogialli, Sara; Chilin, Adriana
Tyrosine kinase inhibitor prodrug-loaded liposomes for controlled release at tumor microenvironment
2021 Salmaso, S.; Mastrotto, F.; Roverso, M.; Gandin, V.; De Martin, S.; Gabbia, D.; De Franco, M.; Vaccarin, C.; Verona, M.; Chilin, A.; Caliceti, P.; Bogialli, S.; Marzaro, G.
Surface plasmon resonance based analysis of the binding of LYAR protein to the rs368698783 (G>A) polymorphic Aγ-globin gene sequences mutated in β-thalassemia
2019 Gemmo, C.; Breveglieri, G.; Marzaro, G.; Lampronti, I.; Cosenza, L. C.; Gasparello, J.; Zuccato, C.; Fabbri, E.; Borgatti, M.; Chilin, A.; Finotti, A.; Gambari, R.
Corilagin Induces High Levels of Apoptosis in the Temozolomide-Resistant T98G Glioma Cell Line
2018 Milani, R; Brognara, E; Fabbri, E; Finotti, A; Borgatti, M; Lampronti, I; Marzaro, Giovanni; Chilin, Adriana; Lee, Kk; Kok, Sh; Chui, Ch; Gambari, R.
Design, synthesis and biological evaluation of novel trimethylangelicin analogues targeting nuclear factor kB (NF-kB)
2018 Marzaro, Giovanni; Lampronti, Ilaria; D'Aversa, Elisabetta; Sacchetti, Gianni; Miolo, Giorgia; Vaccarin, Christian; Cabrini, Giulio; Dechecchi, Maria Cristina; Gambari, Roberto; Chilin, Adriana
Molecular mechanism of action of trimethylangelicin derivatives as CFTR modulators
2018 Laselva, Onofrio; Marzaro, Giovanni; Vaccarin, Christian; Lampronti, Ilaria; Tamanini, Anna; Lippi, Giuseppe; Gambari, Roberto; Cabrini, Giulio; Bear, Christine E.; Chilin, Adriana; Dechecchi, Maria C.
Targeting DNA Binding for NF-κB as an Anticancer Approach in Hepatocellular Carcinoma
2018 Chung, Po-Yee; Lam, Pik-Ling; Zhou, Yuan-Yuan; Gasparello, Jessica; Finotti, Alessia; Chilin, Adriana; Marzaro, Giovanni; Gambari, Roberto; Bian, Zhao-Xiang; Kwok, Wai-Ming; Wong, Wai-Yeung; Wang, Xi; Lam, Alfred King-Yin; Chan, Albert Sun-Chi; Li, Xingshu; Ma, Jessica Yuen-Wuen; Chui, Chung-Hin; Lam, Kim-Hung; Tang, Johnny Cheuk-On
Differential Effects of Angelicin Analogues on NF- κ B Activity and IL-8 Gene Expression in Cystic Fibrosis IB3-1 Cells
2017 Lampronti, Ilaria; Manzione, Maria Giulia; Sacchetti, Gianni; Ferrari, Davide; Spisani, Susanna; Bezzerri, Valentino; Finotti, Alessia; Borgatti, Monica; Dechecchi, Maria Cristina; Miolo, Giorgia; Marzaro, Giovanni; Cabrini, Giulio; Gambari, Roberto; Chilin, Adriana
Discovery of novel wtRET and V804MRET inhibitors: from hit to lead
2017 Mologni, Luca; DALLA VIA, Martina; Chilin, Adriana; Palumbo, Manlio; Marzaro, Giovanni
Investigational drugs targeting cyclin-dependent kinases for the treatment of cancer: an update on recent findings (2013-2016)
2016 Di Giovanni, Carmen; Novellino, Ettore; Chilin, Adriana; Lavecchia, Antonio; Marzaro, Giovanni
Novel benzoquinoline derivatives via unpredicted condensation of ethyl propiolate and naphthylamines: Synthesis and topoisomerase inhibition activity
2016 Marzaro, Giovanni; DALLA VIA, Lisa; GARCIA ARGAEZ, AIDA NELLY; DALLA VIA, Martina; Chilin, Adriana
Structural and Functional Insights on an Uncharacterized Aγ-Globin-Gene Polymorphism Present in Four β(0)-Thalassemia Families with High Fetal Hemoglobin Levels
2016 Bianchi, Nicoletta; Cosenza, Lucia Carmela; Lampronti, Ilaria; Finotti, Alessia; Breveglieri, Giulia; Zuccato, Cristina; Fabbri, Enrica; Marzaro, Giovanni; Chilin, Adriana; De Angelis, Gioia; Borgatti, Monica; Gallucci, Cristiano; Alfieri, Cecilia; Ribersani, Michela; Isgrò, Antonella; Marziali, Marco; Gaziev, Javid; Morrone, Aldo; Sodani, Pietro; Lucarelli, Guido; Gambari, Roberto; Paciaroni, Katia
Substituted quinazolinones as kinase inhibitors endowed with anti-fibrotic properties
2016 Marzaro, Giovanni; Castagliuolo, Ignazio; Schirato, Giulia; Palu', Giorgio; DALLA VIA, Martina; Chilin, Adriana; Brun, Paola