GANDIN, VALENTINA
GANDIN, VALENTINA
Dipartimento di Scienze del Farmaco - DSF
1,3,5-Triaza-7-phosphaadamantane and Cyclohexyl Groups Impart to Di-Iron(I) Complex Aqueous Solubility and Stability, and Prominent Anticancer Activity in Cellular and Animal Models
2024 De Franco, M.; Biancalana, L.; Zappelli, C.; Zacchini, S.; Gandin, V.; Marchetti, F.
Anticancer activity of new water-soluble sulfonated thiosemicarbazone copper(II) complexes targeting disulfide isomerase
2024 Miglioli, F.; De Franco, M.; Bartoli, J.; Scaccaglia, M.; Pelosi, G.; Marzano, C.; Rogolino, D.; Gandin, V.; Carcelli, M.
Anticancer potential of copper(I) complexes based on isopropyl ester derivatives of bis(pyrazol-1-yl)acetate ligands
2024 Pellei, Maura; Santini, Carlo; Caviglia, Miriam; Del Gobbo, Jo'; Battocchio, Chiara; Meneghini, Carlo; Amatori, Simone; Donati, Chiara; Zampieri, Eleonora; Gandin, Valentina; Marzano, Cristina
Palladium(II)-Indenyl Complexes Bearing N-Heterocyclic Carbene (NHC) Ligands as Potent and Selective Metallodrugs toward High-Grade Serous Ovarian Cancer Models
2024 Bortolamiol, E.; Mauceri, M.; Piccolo, R.; Cavarzerani, E.; Demitri, N.; Donati, C.; Gandin, V.; Brezar, S. K.; Kamensek, U.; Cemazar, M.; Canzonieri, V.; Rizzolio, F.; Visentin, F.; Scattolin, T.
Synthesis and Investigations of the Antitumor Effects of First-Row Transition Metal(II) Complexes Supported by Two Fluorinated and Non-Fluorinated β-Diketonates
2024 Pellei, Maura; Del Gobbo, Jo'; Caviglia, Miriam; Gandin, Valentina; Marzano, Cristina; Karade, Deepika V.; Noonikara Poyil, Anurag; Dias, H. V. Rasika; Santini, Carlo
Synthesis, characterization and in vitro cytotoxicity of gallium(iii)-dithiocarbamate complexes
2024 Salvarese, N.; Morellato, N.; Gobbi, C.; Gandin, V.; De Franco, M.; Marzano, C.; Dolmella, A.; Bolzati, C.
Synthesis, structural and computational study, DNA binding and cytotoxic activity of Cu(II) complexes of 6- and 7-chloro-2-oxo-1,2-dihydroquinoline-3-carbaldehyde-2-furoyl-hydrazones
2024 Thirunavukkarasu, Thangavel; Sparkes, Hazel A.; Gandin, Valentina; Marzano, Cristina; Bertani, Roberta; Mozzon, Mirto; Scettri, Anna; Albinati, Alberto; Demartin, Francesco; Casella, Girolamo; Ferrante, Francesco; Zoleo, Alfonso; Sgarbossa, Paolo; Natarajan, Karuppannan
Triiron Complex with N-Ferrocenyl Aminocarbyne Ligand Bridging a Diiron Core: DFT, Electrochemical, and Biological Insights
2024 Saviozzi, Chiara; Biancalana, Lorenzo; Funaioli, Tiziana; Bortoluzzi, Marco; De Franco, Michele; Guelfi, Massimo; Gandin, Valentina; Marchetti, Fabio
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
2023 Pecoraro, Camilla; DE FRANCO, Michele; Carbone, Daniela; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall'Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; DE FRANCO, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Multitargeting Prodrugs that Release Oxaliplatin, Doxorubicin and Gemcitabine are Potent Inhibitors of Tumor Growth and Effective Inducers of Immunogenic Cell Death
2023 Sarkar, Amrita; Novohradsky, Vojtech; Maji, Moumita; Babu, Tomer; Markova, Lenka; Kostrhunova, Hana; Kasparkova, Jana; Gandin, Valentina; Brabec, Viktor; Gibson, Dan
Novel Biotinylated Cu(II)-Phenanthroline Complexes: 2D and 3D Cytotoxic Activity and Mechanistic Insight
2023 Barrett, Stephen; De Franco, Michele; Donati, Chiara; Marzano, Cristina; Gandin, Valentina; Montagner, Diego
Novel design of dual-action Pt(iv) anticancer pro-drugs based on cisplatin and derivatives of the tyrosine kinase inhibitors imatinib and nilotinib
2023 Beirne, Darren Fergal; Farkaš, Barbara; Donati, Chiara; Gandin, Valentina; Rozas, Isabel; Velasco-Torrijos, Trinidad; Montagner, Diego
Novel Silver Complexes Based on Phosphanes and Ester Derivatives of Bis(pyrazol-1-yl)acetate Ligands Targeting TrxR: New Promising Chemotherapeutic Tools Relevant to SCLC Management
2023 Pellei, Maura; Santini, Carlo; Bagnarelli, Luca; Caviglia, Miriam; Sgarbossa, Paolo; De Franco, Michele; Zancato, Mirella; Marzano, Cristina; Gandin, Valentina
Oral Anticancer Heterobimetallic PtIV−AuIComplexes Show High In Vivo Activity and Low Toxicity
2023 Babu, Tomer; Ghareeb, Hiba; Basu, Uttara; Schueffl, Hemma; Theiner, Sarah; Heffeter, Petra; Koellensperger, Gunda; Metanis, Norman; Gandin, Valentina; Ott, Ingo; Schmidt, Claudia; Gibson, Dan
Pt(ii) and Pt(iv) complexes with a major component of royal jelly as innovative antitumor drug candidates
2023 Barbanente, Alessandra; Gandin, Valentina; Donati, Chiara; Pierro, Carmela Ilaria; Natile, Giovanni; Margiotta, Nicola
Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma
2023 Carbone, Daniela; De Franco, Michele; Pecoraro, Camilla; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall’Acqua, Stefano; Sut, Stefania; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
Synthesis and cytotoxicity studies of Cu(i) and Ag(i) complexes based on sterically hindered β-diketonates with different degrees of fluorination
2023 Pellei, Maura; Del Gobbo, Jo’; Caviglia, Miriam; Karade, Deepika V.; Gandin, Valentina; Marzano, Cristina; Noonikara Poyil, Anurag; Dias, H. V. Rasika; Santini, Carlo
Unusual tellurium(iv) mediated cyclisation diols into dihydroxazoles with potential anticancer activity
2023 D’Arcy, Kenneth; Schäfer, Tim; De Franco, Michele; Ricco, Raffaele; Gandin, Valentina; Sanz Miguel, Pablo J.; Montagner, Diego
Antiproliferative activity of nickel(II), palladium(II) and zinc(II) thiosemicarbazone complexes
2022 Carcelli, M.; Montalbano, S.; Rogolino, D.; Gandin, V.; Miglioli, F.; Pelosi, G.; Buschini, A.