CARTA, DAVIDE
CARTA, DAVIDE
Dipartimento di Scienze del Farmaco - DSF
99mTc(N)-DBODC(5), a potential radiolabeled probe for SPECT of multidrug resistance: in vitro study
2013 Bolzati, Cristina; Carta, Davide; Gandin, Valentina; Marzano, Cristina; Morellato, Nicolo'; Salvarese, Nicola; M., Cantore; N. A., Colabufo
[99mTc(N)(DBODC)(5)]+: sub-cellular distribution and metabolism studies of this new potential myocardial imaging agent
2009 Bolzati, Cristina; M., CAVAZZA CECCATO; F., Refosco; S., Tokunaga; Salvarese, Nicola; Carta, Davide; Dolmella, Alessandro; Casara, Dario; Bandoli, Giuliano
[Re-188(N)(cys similar to)(PNP)](+/0) mixed ligand compounds as models for target specific agents
2010 Bolzati, Cristina; Thieme, S; Agostini, S; Carta, Davide; Salvarese, Nicola; Refosco, F; Bergmann, R; Pietzsch, J; Pietzsch, Hj
Amidic Coupling in the Synthesis of Pyrroloquinoline 4- and 9-Carboxamides as Potential STAT3 Inhibitors
2018 Carta, Davide; Dal Prà, Matteo; Grazia Ferlin, Maria
An overview on 2-arylquinolin-4(1h)-ones and related structures as tubulin polymerisation inhibitors
2014 Carta, Davide; Ferlin, MARIA GRAZIA
Assessment of the best N3− donors in preparation of [M(N)(PNP)]-based (M=99mTc-; 188Re) target-specific radiopharmaceuticals: Comparison among succinic dihydrazide (SDH), N-methyl-S-methyl dithiocarbazate (HDTCZ) and PEGylated N-methyl-S-methyl dithiocarbazate (HO2C-PEG600-DTCZ)
2014 Carta, Davide; Christian, Jentschel; Stefan, Thieme; Salvarese, Nicola; Nicolò, Morellato; Fiorenzo, Refosco; Paolo, Ruzza; Ralf, Bergmann; Hans Jurgen, Pietzsch; Bolzati, Cristina
Avidin–biotin system: a small library of cysteine biotinylated derivativesdesigned for the [99mTc(N)(PNP)]2+ metal fragment
2006 C., Bolzati; Caporale, Andrea; Agostini, Stefania; Carta, Davide; M., Cavazza Ceccato; F., Refosco; Tisato, F. r.; Schievano, Elisabetta; Bandoli, Giuliano
Biological in vitro and in vivo studies of a series of new asymmetrical cationic [99mTc(N)(DTC-Ln)(PNP)]+ complex (DTC-Ln = alicyclic dithiocarbamate, PNP = diphosphinoamine)
2010 C., Bolzati; M., CAVAZZA CECCATO; S., Agostini; F., Refosco; Y., Yamamichi; S., Tokunaga; Carta, Davide; Salvarese, Nicola; Bernardini, Daniele; Bandoli, Giuliano
Chelating Systems for 99mTc/188Re in the Development of Radiolabeled Peptide Pharmaceuticals
2012 Bolzati, Cristina; Carta, Davide; Salvarese, Nicola; Fiorenzo, Refosco
Design, synthesis, and photophysical properties of pyrroloquinoline-based compounds showing strong blue fluorescence as potential dyes for biomedical applications
2015 Carta, Davide; Balasso, Anna; Caliceti, Paolo; Ferlin, MARIA GRAZIA
Design, Synthesis, and Structure–Activity Relationships of Azolylmethylpyrroloquinolines as Nonsteroidal Aromatase Inhibitors
2013 Ferlin, MARIA GRAZIA; Carta, Davide; Bortolozzi, Roberta; Razieh, Ghodsi; Adele, Chimento; Vincenzo, Pezzi; Moro, Stefano; Nina, Hanke; Rolf W., Hartmann; Basso, Giuseppe; Viola, Giampietro
EB-3D a novel choline kinase inhibitor induces deregulation of the AMPK-mTOR pathway and apoptosis in leukemia T-cells
2018 Mariotto, Elena; Bortolozzi, Roberta; Volpin, Ilaria; Carta, Davide; Serafin, Valentina; Accordi, Benedetta; Basso, Giuseppe; Navarro, Pilar Luque; López-Cara, Luisa Carlota; Viola, Giampietro
Evaluating the effects of fluorine on biological properties and metabolic stability of some antitubulin 3-substituted 7-phenyl-pyrroloquinolinones
2019 Bortolozzi, R.; Carta, D.; Dal Pra, M.; Antoniazzi, G.; Mattiuzzo, E.; Sturlese, M.; Di Paolo, V.; Calderan, L.; Moro, S.; Hamel, E.; Quintieri, L.; Ronca, R.; Viola, G.; Ferlin, M. G.
Insights into the failure of the potential, neutral myocardial imaging agent TcN-NOET: physicochemical identification of by-products and degradation species
2012 Francesco, Tisato; Bolzati, Cristina; Fiorenzo, Refosco; Marina, Porchia; Roberta, Seraglia; Carta, Davide; Roberto, Pasqualini
Melanoma targeting with [99mTc(N)(PNP3)]-labeled α-melanocyte stimulating hormone peptide analogs: Effects of cyclization on the radiopharmaceutical properties
2016 Carta, Davide; Salvarese, Nicola; Morellato, Nicolo'; Gao, Feng; Sihver, Wiebke; Pietzsch, Hans Jurgen; Biondi, Barbara; Ruzza, Paolo; Refosco, Fiorenzo; Carpanese, Debora; Rosato, Antonio; Bolzati, Cristina
Method for optimizing coating properties based on an evolutionary algorithm approach
2011 Carta, Davide; Villanova, Laura; Costacurta, Stefano; Patelli, Alessandro; Poli, Irene; Vezzu', Simone; Scopece, Paolo; Lisi, Fabio; Smith Miles, Kate; Hyndman, Rob J.; Hill, Anita J.; Falcaro, Paolo
Novel 3-Substituted 7-Phenylpyrrolo[3,2-f]quinolin-9(6H)-ones as Single Entities with Multitarget Antiproliferative Activity
2015 Carta, Davide; Bortolozzi, Roberta; Hamel, Ernest; Basso, Giuseppe; Moro, Stefano; Viola, Giampietro; Ferlin, MARIA GRAZIA
Peroxisome proliferator-activated receptor-γ mediates the anti-inflammatory effect of 3-hydroxy-4-pyridinecarboxylic acid derivatives: Synthesis and biological evaluation
2013 Brun, Paola; Dean, Annalisa; DI MARCO, Valerio; P., Surajit; Castagliuolo, Ignazio; Carta, Davide; Ferlin, MARIA GRAZIA
Pharmacological characterization of α-MSH-derivatives
2014 Sihver, W.; Gao, F.; Jurischka, C.; Haase Kohn, C.; Steinbach, J.; Carta, Davide; Bolzati, Cristina; Calderan, Andrea; Pietzsch, J.; Pietzsch, H. J.
Radiopharmacological characterization of 64Cu-labeled α-MSH analogs for potential use in imaging of malignant melanoma
2016 Gao, Feng; Sihver, Wiebke; Jurischka, Christoph; Bergmann, Ralf; Haase Kohn, Cathleen; Mosch, Birgit; Steinbach, Jörg; Carta, Davide; Bolzati, Cristina; Calderan, Andrea; Pietzsch, Jens; Pietzsch, Hans Jürgen