BORTOLOZZI, ROBERTA
BORTOLOZZI, ROBERTA
Dipartimento di Scienze del Farmaco - DSF
A first-in-class Wiskott-Aldrich syndrome protein activator with anti-tumor activity in hematologic cancers
2024 Spriano, Filippo; Sartori, Giulio; Sgrignani, Jacopo; Barnabei, Laura; Arribas, Alberto J; Guala, Matilde; Del Amor, Ana Maria Carrasco; Tomasso, Meagan R; Tarantelli, Chiara; Cascione, Luciano; Golino, Gaetanina; Riveiro, Maria E; Bortolozzi, Roberta; Lupia, Antonio; Paduano, Francesco; Huguet, Samuel; Rezai, Keyvan; Rinaldi, Andrea; Margheriti, Francesco; Ventura, Pedro; Guarda, Greta; Costa, Giosuè; Rocca, Roberta; Furlan, Alberto; Verdonk, Luuk M; Innocenti, Paolo; Martin, Nathaniel I; Viola, Giampietro; Driessen, Christoph; Zucca, Emanuele; Stathis, Anastasios; Gahtory, Digvijay; Van den Nieuwboer, Maurits; Bornhauser, Beat; Alcaro, Stefano; Trapasso, Francesco; Cristobal, Susana; Padrick, Shae B; Pazzi, Natalina; Cavalli, Franco; Cavalli, Andrea; Gaudio, Eugenio; Bertoni, Francesco
A Multi-Omics Approach Reveals Enrichment in Metabolites Involved in the Regulation of the Glutathione Pathway in LIN28B-Dependent Cancer Cells
2024 Stocchero, Matteo; Corallo, Diana; Bresolin, Silvia; Pantile, Marcella; Pirillo, Paola; Bortolozzi, Roberta; Menegazzo, Sara; Boso, Daniele; Viola, Giampietro; Baraldi, Eugenio; Biffi, Alessandra; Giordano, Giuseppe; Aveic, Sanja
Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold
2023 Romagnoli, Romeo; De Ventura, Tiziano; Manfredini, Stefano; Baldini, Erika; Supuran, Claudiu T; Nocentini, Alessio; Brancale, Andrea; Bortolozzi, Roberta; Manfreda, Lorenzo; Viola, Giampietro
Identification of Homoharringtonine as a potent inhibitor of glioblastoma cell proliferation and migration
2023 Porcù, Elena; Maule, Francesca; Manfreda, Lorenzo; Mariotto, Elena; Bresolin, Silvia; Cani, Alice; Bortolozzi, Roberta; Puppa, Alessandro Della; Corallo, Diana; Viola, Giampietro; Rampazzo, Elena; Persano, Luca
Identification of pyrrolo[3',4':3,4]cyclohepta[1,2-d][1,2]oxazoles as promising new candidates for the treatment of lymphomas
2023 Barreca, Marilia; Spanò, Virginia; Rocca, Roberta; Bivacqua, Roberta; Gualtieri, Gianmarco; Raimondi, Maria Valeria; Gaudio, Eugenio; Bortolozzi, Roberta; Manfreda, Lorenzo; Bai, Ruoli; Montalbano, Alessandra; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Viola, Giampietro; Barraja, Paola
Molecular and functional profiling of chemotolerant cells unveils nucleoside metabolism-dependent vulnerabilities in medulloblastoma
2023 Mariotto, Elena; Rampazzo, Elena; Bortolozzi, Roberta; Rruga, Fatlum; Zeni, Ilaria; Manfreda, Lorenzo; Marchioro, Chiara; Canton, Martina; Cani, Alice; Magni, Ruben; Luchini, Alessandra; Bresolin, Silvia; Viola, Giampietro; Persano, Luca
Surviving the hunger games: Metabolic reprogramming in medulloblastoma
2023 Manfreda, Lorenzo; Rampazzo, Elena; Persano, Luca; Viola, Giampietro; Bortolozzi, Roberta
Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis
2022 Romagnoli, R.; Oliva, P.; Prencipe, F.; Manfredini, S.; Germano, M. P.; De Luca, L.; Ricci, F.; Corallo, D.; Aveic, S.; Mariotto, E.; Viola, G.; Bortolozzi, R.
Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities
2022 Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Budassi, Federica; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Manfreda, Lorenzo; Mariotto, Elena; Bortolozzi, Roberta; Viola, Giampietro
Histone Deacetylase Inhibitors Impair Glioblastoma Cell Motility and Proliferation
2022 Rampazzo, E.; Manfreda, L.; Bresolin, S.; Cani, A.; Mariotto, E.; Bortolozzi, R.; Della Puppa, A.; Viola, G.; Persano, L.
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
2022 Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Synthesis of 2H-Imidazo[2′,1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations
2022 Cilibrasi, V.; Spano, V.; Bortolozzi, R.; Barreca, M.; Raimondi, M. V.; Rocca, R.; Maruca, A.; Montalbano, A.; Alcaro, S.; Ronca, R.; Viola, G.; Barraja, P.
A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents
2021 Romagnoli, R.; Oliva, P.; Salvador, M. K.; Manfredini, S.; Padroni, C.; Brancale, A.; Ferla, S.; Hamel, E.; Ronca, R.; Maccarinelli, F.; Rruga, F.; Mariotto, E.; Viola, G.; Bortolozzi, R.
Concise synthesis and biological evaluation of 2-Aryl-3-Anilinobenzo[b]thiophene derivatives as potent apoptosis-inducing agents
2021 Romagnoli, R.; Preti, D.; Hamel, E.; Bortolozzi, R.; Viola, G.; Brancale, A.; Ferla, S.; Morciano, G.; Pinton, P.
Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems
2021 Grieco, I.; Bissaro, M.; Tiz, D. B.; Perez, D. I.; Perez, C.; Martinez, A.; Redenti, S.; Mariotto, E.; Bortolozzi, R.; Viola, G.; Cozza, G.; Spalluto, G.; Moro, S.; Federico, S.
Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors
2021 Spano, V.; Barreca, M.; Rocca, R.; Bortolozzi, R.; Bai, R.; Carbone, A.; Raimondi, M. V.; Piccionello, A. P.; Montalbano, A.; Alcaro, S.; Hamel, E.; Viola, G.; Barraja, P.
Synthesis, DNA-binding and antiproliferative properties of diarylquinolizinium derivatives
2021 Bortolozzi, Roberta; Ihmels, Heiko; Schulte, Robin; Stremmel, Christopher; Viola, Giampietro
Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization
2020 Romagnoli, R.; Prencipe, F.; Oliva, P.; Kimatrai Salvador, M.; Brancale, A.; Ferla, S.; Hamel, E.; Viola, G.; Bortolozzi, R.; Persoons, L.; Balzarini, J.; Liekens, S.; Schols, D.
Design, synthesis, in vitro and in vivo biological evaluation of 2-amino-3-aroylbenzo[b]furan derivatives as highly potent tubulin polymerization inhibitors
2020 Oliva, Paola; Romagnoli, Romeo; Manfredini, Stefano; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Maccarinelli, Federica; Giacomini, Arianna; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Ecdysteroid Derivatives that Reverse P-Glycoprotein-Mediated Drug Resistance
2020 Bortolozzi, R.; Luraghi, A.; Mattiuzzo, E.; Sacchetti, A.; Silvani, A.; Viola, G.