MEGGIO, FLAVIO
MEGGIO, FLAVIO
Inhibition of Protein Kinase CK2 by Flavonoids and Tyrphostins. A Structural Insight.
2012 Lolli, Graziano; Cozza, Giorgio; Mazzorana, Marco; Tibaldi, Elena; Cesaro, Luca; Donella, Arianna; Meggio, Flavio; Venerando, Andrea; Franchin, Cinzia; Sarno, Stefania; Battistutta, Roberto; Pinna, Lorenzo
Structural features underlying the selectivity of the kinase inhibitors NBC and dNBC: role of a nitro group that discriminates between CK2 and DYRK1A
2012 Sarno, Stefania; Mazzorana, Marco; Ryan, Traynor; Ruzzene, Maria; Cozza, Giorgio; Pagano, MARIO ANGELO PRIMO; Meggio, Flavio; Zagotto, Giuseppe; Battistutta, Roberto; Pinna, Lorenzo
ATP Site-Directed Inhibitors of Protein Kinase CK2: An Update
2011 Sarno, Stefania; Papinutto, Elena; Franchin, Cinzia; Bain, J; Elliott, M; Meggio, Flavio; Kazimierczuk, Z; Orzeszko, A; Zanotti, Giuseppe; Battistutta, Roberto; Pinna, Lorenzo
The Dark Side of Protein Kinase CK2 Inhibition
2011 Cozza, Giorgio; Meggio, Flavio; Moro, Stefano
Understanding protein kinase CK2 mis-regulation upon F508del CFTR expression
2011 Venerando, Andrea; Pagano, MARIO ANGELO PRIMO; Tosoni, Kendra; Meggio, Flavio; Diane, Cassidy; Michelle, Stobbart; Pinna, Lorenzo; Anil, Mehta
Unprecedented Selectivity and Structural Determinants of a New Class of Protein Kinase CK2 Inhibitors in Clinical Trials for the Treatment of Cancer
2011 Battistutta, Roberto; Cozza, Giorgio; F., Pierre; Papinutto, Elena; Lolli, Graziano; Sarno, Stefania; S. E., O'Brien; A., Siddiqui Jain; M., Haddach; K., Anderes; D. M., Ryckman; Meggio, Flavio; Pinna, Lorenzo
Urolithin as a converging scaffold linking ellagic acid and coumarin analogues: design of potent protein kinase CK2 inhibitors.
2011 Cozza, Giorgio; Gianoncelli, Alessandra; Bonvini, Paolo; Zorzi, Elisa; Pasquale, Riccardo; Rosolen, Angelo; Pinna, Lorenzo; Meggio, Flavio; Zagotto, Giuseppe; Moro, Stefano
Cystic fibrosis transmembrane regulator fragments with the Phe508 deletion exert a dual allosteric control over the master kinase CK2
2010 Pagano, MARIO ANGELO PRIMO; Marin, Oriano; Cozza, Giorgio; Sarno, Stefania; Meggio, Flavio; Treharne, Kj; Mehta, A; Pinna, Lorenzo
Pancreatic and duodenal homeobox 1 (PDX1) phosphorylation at serine-269 is HIPK2-dependent and affects PDX1 subnuclear localization
2010 An, R; Xavier, Gd; Semplici, F; Vakhshouri, S; Hao, Hx; Rutter, J; Pagano, Ma; Meggio, Flavio; Pinna, Lorenzo; Rutter, Ga
The pleiotropic protein kinase CK2 phosphorylates HTLV-1 Tax protein in vitro, targeting its PDZ-binding motif
2010 Bidoia, C; Mazzorana, M; Pagano, MARIO ANGELO PRIMO; Arrigoni, Giorgio; Meggio, Flavio; Pinna, Lorenzo; Bertazzoni, U.
A Modified KESTREL Search Reveals a Basophilic Substrate Consensus for the Saccharomyces cerevisiae Npr1 Protein Kinase
2009 Gander, S; Martin, D; Hauri, S; Moes, S; Poletto, G; Pagano, MARIO ANGELO PRIMO; Marin, Oriano; Meggio, Flavio; Jenoe, P.
Cystic fibrosis transmembrane regulator fragments with the Phe508 deletion exert a dual allosteric control over the master kinase CK2.
2009 Pagano, Ma; Marin, Oriano; Cozza, Giorgio; Sarno, Stefania; Meggio, Flavio; Treharne, Kj; Mehta, A; Pinna, La
Identification of new powerful and selectiveinhibitors of protein kinases CK1δ and CK2 bycomputer aided virtual screening and molecularderivatization of anthraquinone scaffolds
2009 Cozza, Giorgio; Gianoncelli, A; Venerando, Andrea; DI MAIRA, Giovanni; Montopoli, Monica; Sarno, Stefania; Ruzzene, Maria; Pagano, MARIO ANGELO PRIMO; Moro, Stefano; Caparrotta, Laura; Zagotto, Giuseppe; Pinna, Lorenzo; Meggio, Flavio
Quinalizarin as a potent, selective and cell-permeable inhibitor of protein kinase CK2
2009 Cozza, Giorgio; Mazzorana, Marco; Papinutto, Elena; Bain, J; Elliott, M; DI MAIRA, Giovanni; Gianoncelli, Alessandra; Pagano, MARIO ANGELO PRIMO; Sarno, Stefania; Ruzzene, Maria; Battistutta, Roberto; Meggio, Flavio; Moro, Stefano; Zagotto, Giuseppe; Pinna, La
Scouting Novel Protein Kinase A (PKA) Inhibitors by Using a Consensus Docking-Based Virtual Screening Approach
2009 Zonta, N; Cozza, Giorgio; Gianoncelli, Alessandra; Korb, O; Exner, Te; Meggio, Flavio; Zagotto, Giuseppe; Moro, Stefano
Tetraiodobenzimidazoles are potent inhibitors of protein kinase CK2
2009 Gianoncelli, A; Cozza, Giorgio; Orzeszko, A; Meggio, Flavio; Kazimierczuk, Z; Pinna, Lorenzo
Coumarin as attractive casein kinase 2(CK2) inhibitor scaffold: an integrated approach to elucidate the putative binding motif and explain structure-activity relationship.
2008 Chilin, Adriana; Battistutta, Roberto; Bortolato, Andrea; Cozza, Giorgio; Zanatta, Samuele; Poletto, G; Mazzorana, Marco; Zagotto, Giuseppe; Uriarte, E; Guiotto, Adriano; Pinna, Lorenzo; Meggio, Flavio; Moro, Stefano
Identification of novel protein kinase CK1 delta (CK1 delta) inhibitors through structure-based virtual screening
2008 Cozza, Giorgio; Gianoncelli, A; Montopoli, Monica; Caparrotta, Laura; Venerando, Andrea; Meggio, Flavio; Pinna, Lorenzo; Zagotto, Giuseppe; Moro, Stefano
Modulation of protein kinase CK2 activity by fragments of CFTR encompassing F508 may reflect functional links with cystic fibrosis pathogenesis
2008 Pagano, MARIO ANGELO PRIMO; Arrigoni, Giorgio; Marin, Oriano; Sarno, Stefania; Meggio, Flavio; Treharne, Kj; Mehta, A; Pinna, Lorenzo
Regulatory subunit of protein kinase CK2 contributes to the recognition of the substrate consensus sequence. A study with an eIF2 beta-derived peptide
2008 Poletto, Giorgia; Vilardell, J; Marin, Oriano; Pagano, Ma; Cozza, Giorgio; Sarno, Stefania; Falques, A; Itarte, E; Pinna, Lorenzo; Meggio, Flavio