BATTISTUTTA, ROBERTO
BATTISTUTTA, ROBERTO
Dipartimento di Scienze Chimiche - DiSC
Allostery in homodimeric SARS-CoV-2 main protease
2024 Fornasier, Emanuele; Fabbian, Simone; Shehi, Haidi; Enderle, Janine; Gatto, Barbara; Volpin, Daniele; Biondi, Barbara; Bellanda, Massimo; Giachin, Gabriele; Sosic, Alice; Battistutta, Roberto
One substrate many enzymes virtual screening uncovers missing genes of carnitine biosynthesis in human and mouse
2024 Malatesta, M.; Fornasier, E.; Di Salvo, M. L.; Tramonti, A.; Zangelmi, E.; Peracchi, A.; Secchi, A.; Polverini, E.; Giachin, G.; Battistutta, R.; Contestabile, R.; Percudani, R.
A new inactive conformation of SARS-CoV-2 main protease
2022 Fornasier, Emanuele; Macchia, Maria Ludovica; Giachin, Gabriele; Sosic, Alice; Pavan, Matteo; Sturlese, Mattia; Salata, Cristiano; Moro, Stefano; Gatto, Barbara; Bellanda, Massimo; Battistutta, Roberto
Computationally driven discovery of SARS-CoV-2 Mpro inhibitors: from design to experimental validation
2022 El Khoury, Léa; Jing, Zhifeng; Cuzzolin, Alberto; Deplano, Alessandro; Loco, Daniele; Sattarov, Boris; Hédin, Florent; Wendeborn, Sebastian; Ho, Chris; El Ahdab, Dina; Jaffrelot-Inizan, Theo; Sturlese, M; Sosic, Alice; Volpiana, Martina; Lugato, Angela; Barone, Marco; Gatto, Barbara; Macchia, Maria Ludovica.; Bellanda, M; Battistutta, Roberto; Salata, Cristiano; Kondratov, Ivan; Iminov, Rustan; Khairulin, Andrii; Mykhalonok, Yaroslav; Pochepko, Anton; Chashka-Ratushnyi, Volodymyr; Kos, Iaroslava; Moro, Stefano; Montes, Matthieu; Ren, Pengyu; Ponder, Jay W.; Lagardère, Louis; Piquemal, Jean-Philip; Sabbadin, Davide
IDENTIFICATION OF NEW SARS-COV-2 MAIN PROTEASE INHIBITORS BY AN INTEGRATED IN-SILICO AND IN-VITRO STRATEGY
2022 Salata, C.; Mirandola, M.; Salaris, C.; Macchia, M. L.; Fornasier, E.; Pavan, M.; Giachin, G.; Sosic, A.; Sturlese, M.; Bellanda, M.; Battistutta, R.; Moro, S.; Gatto, B.
Mechanism of CK2 Inhibition by a Ruthenium-Based Polyoxometalate
2022 Fabbian, S; Giachin, G; Bellanda, M; Borgo, C; Ruzzene, M; Spuri, G; Campofelice, A; Veneziano, L; Bonchio, M; Carraro, M; Battistutta, R
Calmodulin binds to the STAS domain of SLC26A5 prestin with a calcium-dependent, one-lobe, binding mode
2021 Costanzi, E.; Coletti, A.; Zambelli, B.; Macchiarulo, A.; Bellanda, M.; Battistutta, R.
Comparative molecular dynamics investigation of the electromotile hearing protein prestin
2021 Abrusci, G.; Tarenzi, T.; Sturlese, M.; Giachin, G.; Battistutta, R.; Lattanzi, G.
A novel class of selective CK2 inhibitors targeting its open hinge conformation
2020 Dalle Vedove, Andrea; Zontab, Francesca; Zanforlin, Enrico; Demitri, Nicola; Ribaudo, Giovanni; Cazzanelli, Giulia; Ongaro, Alberto; Sarno, Stefania; Zagotto, Giuseppe; Battistutta, Roberto; Ruzzene, Maria; Lolli, Graziano
Biochemical and cellular mechanism of protein kinase CK2 inhibition by deceptive curcumin
2020 Cozza, Giorgio; Zonta, Francesca; Dalle Vedove, Andrea; Venerando, Andrea; Dall'Acqua, Stefano; Battistutta, Roberto; Ruzzene, Maria; Lolli, Graziano
Axonal Odorant Receptors Mediate Axon Targeting
2019 Zamparo, I.; Francia, S.; Franchi, S. A.; Redolfi, N.; Costanzi, E.; Kerstens, A.; Fukutani, Y.; Battistutta, R.; Polverino de Laureto, P.; Munck, S.; De Strooper, B.; Matsunami, H.; Lodovichi, C.
Inhibitory Properties of ATP-Competitive Coumestrol and Boldine Are Correlated to Different Modulations of CK2 Flexibility
2019 Battistutta, R.; Lolli, G.
Insight into GFPmut2 pH Dependence by Single Crystal Microspectrophotometry and X-ray Crystallography
2018 Lolli, Graziano; Raboni, Samanta; Pasqualetto, Elisa; Benoni, Roberto; Campanini, Barbara; Ronda, Luca; Mozzarelli, Andrea; Bettati, Stefano; Battistutta, Roberto
Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR
2018 Carlino, Luca; Christodoulou, Michael S.; Restelli, Valentina; Caporuscio, Fabiana; Foschi, Francesca; Semrau, Marta S.; Costanzi, Elisa; Tinivella, Annachiara; Pinzi, Luca; Lo Presti, Leonardo; Battistutta, Roberto; Storici, Paola; Broggini, Massimo; Passarella, Daniele; Rastelli, Giulio
Characterization of the oligomeric states of the CK2 alpha2beta2 holoenzyme in solution
2017 Lolli, Graziano; Naressi, Denise; Sarno, Stefania; Battistutta, Roberto
Identification and characterization of three novel mutations in the CASQ1 gene in four patients with tubular aggregate myopathy
2017 Barone, Virginia; Del Re, Valeria; Gamberucci, Alessandra; Polverino, Valentina; Galli, Lucia; Rossi, Daniela; Costanzi, Elisa; Toniolo, Luana; Berti, Gianna; Malandrini, Alessandro; Ricci, Giulia; Siciliano, Gabriele; Vattemi, Gaetano; Tomelleri, Giuliano; Pierantozzi, Enrico; Spinozzi, Simone; Volpi, Nila; Fulceri, Rosella; Battistutta, Roberto; Reggiani, Carlo; Sorrentino, Vincenzo
Probing an Allosteric Pocket of CDK2 with Small Molecules
2017 Christodoulou, Michael S.; Caporuscio, Fabiana; Restelli, Valentina; Carlino, Luca; Cannazza, Giuseppe; Costanzi, Elisa; Citti, Cinzia; Lo Presti, Leonardo; Pisani, Pasquale; Battistutta, Roberto; Broggini, Massimo; Passarella, Daniele; Rastelli, Giulio
The STAS domain of mammalian SLC26A5 prestin harbours an anion-binding site
2016 Lolli, Graziano; Pasqualetto, Elisa; Costanzi, Elisa; Bonetto, Greta; Battistutta, Roberto
Structural basis of CK2 regulation by autoinhibitory oligomerization
2015 Lolli, G.; Battistutta, R.
Active Form of the Protein Kinase CK2 alpha(2)beta(2) holoenzyme Is a Strong Complex with Symmetric Architecture
2014 Lolli, Graziano; Ranchio, Alessandro; Battistutta, Roberto